平安! 发表于 2011-11-9 19:57 2 B' |! J# r# M, U0 y
Pazopanib (100 mg/kg/day free base equivalent)
H8 k$ f' N% {" f& @0 c: X0 W7 l 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。4 G8 `8 g1 C T5 G
搜索了一下,原料一大堆。
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7 n0 `) I( Z) H/ r$ D对不起!100mg/kg是用于移植瘤的,我弄错了。
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$ n, d" N, l: G; K- e6 g" O以下是正版说明书的推荐用量。: N& U& d5 c+ m9 e! ~1 F
9 r4 b3 D7 A! ^% D+ h8 ~! U--------------------- DOSAGE AND ADMINISTRATION ----------------' W! Y6 T( S }' U4 z5 b x. [
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
5 a5 s- z- N" }) N D/ J9 L6 h* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) . a: q/ p5 ^& n$ C9 m) J3 M
---------------------DOSAGE FORMS AND STRENGTHS --------------8 o' A6 U g6 D4 `+ @- H, @' D
200 mg tablets. (3) 2 B' }) O+ U6 D3 E, R
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